RESEARCH IN CHEMICAL SCIENCES (CS)

2020

Updated on January 28, 2021

1. An anticonvulsive drug, valproic acid (valproate), has effects on the biosynthesis of fatty acids and polyketides in microorganisms

By: Poolchanuan, P., Unagul, P., Thongnest, S., Wiyakrutta, S., Ngamrojanavanich, N., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Scientific Reports
Vol.: 10
No.: 1
Page:
Published: 2020
doi: https://doi.org/10.1038/s41598-020-66251-y

2. Antifungal activity of 8-methoxynaphthalen-1-ol isolated from the endophytic fungus Diatrype palmicola MFLUCC 17-0313 against the plant pathogenic fungus Athelia rolfsii on tomatoes

By: Tanapichatsakul, C., Pansanit, A., Monggoot, S., Brooks, S., Prachya, S., Kittakoop, P., Panuwet, P., and Pripdeevech, P.
PeerJ
Vol.: 8
No.:
Page:
Published: 2020
doi: https://doi.org/10.7717/peerj.9103

3. Antioxidant and acetylcholinesterase inhibitory activities of Morinda citrifolia L. extracts

By: Sam-ang, P., Surangkul, D., Savaspun, K., and Phanumartwiwath, A.
Agriculture and Natural Resources
Vol.: 54
No.: 2
Page: 173–179
Published: 2020
doi:

4. Atalantiaphyllines A-G, prenylated acridones from Atalantia monophylla DC. and their aromatase inhibition and cytotoxic activities

By: Pailee, P., Prawat, H., Ploypradith, P., Mahidol, C., Ruchirawat, S., and Prachyawarakorn, V.
Phytochemistry
Vol.: 180
No.:
Page:
Published: 2020
doi: https://doi.org/10.1016/j.phytochem.2020.112525

5. Biscurcudiols, myrmekioperoxides, and myrmekiodermaral from the Thai marine sponge Myrmekioderma sp.

By: Wongbundit, S., Mahidol, C., Kaweetripob, W., Prachyawarakorn, V., Eurtivong, C., Sahakitpichan, P., Tuntiwachwuttikul, P., Ruchirawat, S., and Prawat, H.
Tetrahedron
Vol.: 76
No.: 19
Page:
Published: 2020
doi: https://doi.org/10.1016/j.tet.2020.131162

6. Chemoselective acid-catalyzed 4+2 -cycloaddition reactions of ortho-quinone methides and styrenes/stilbenes/cinnamates

By: Akkarasereenon, K., Tangdenpaisal, K., Ruchirawat, S., and Ploypradith, P.
Organic & Biomolecular Chemistry
Vol.: 18
No.: 43
Page: 8854-8866
Published: 2020
doi: https://doi.org/10.1039/d0ob01312a

7. Commercial Copper-Catalyzed Aerobic Oxidative Synthesis of Quinazolinones from 2-Aminobenzamide and Methanol

By: Kerdphon, S., Sanghong, P., Chatwichien, J., Choommongkol, V., Rithchumpon, P., Singh, T., and Meepowpan, P.
European Journal of Organic Chemistry
Vol.: 2020
No.: 18
Page: 2730-2734
Published: 2020
doi: https://doi.org/10.1002/ejoc.202000257

8. Discovery of New and Potent InhA Inhibitors as Antituberculosis Agents: Structure-Based Virtual Screening Validated by Biological Assays and X-ray Crystallography

By: Kamsri, P., Hanwarinroj, C., Phusi, N., Pornprom, T., Chayajarus, K., Punkvang, A., Suttipanta, N., Srimanote, P., Suttisintong, K., Songsiriritthigul, C., Saparpakorn, P., Hannongbua, S., Rattanabunyong, S., Seetaha, S., Choowongkomon, K., Sureram, S., Kittakoop, P., Hongmanee, P., Santanirand, P., Chen, Z. Q., Zhu, W. L., Blood, R. A., Takebayashi, Y., Hinchliffe, P., Mulholland, A. J., Spencer, J., and Pungpo, P.
Journal of Chemical Information and Modeling
Vol.: 60
No.: 1
Page: 226-234
Published: 2020
doi: https://doi.org/10.1021/acs.jcim.9b00918

9. Discovery of novel halogenated 8-hydroxyquinoline-based anti-MRSA agents: In vitro and QSAR studies

By: Cherdtrakulkiat, R., Worachartcheewan, A., Tantimavanich, S., Lawung, R., Sinthupoom, N., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Drug Development Research
Vol.: 81
No.: 1
Page: 127-135
Published: 2020
doi: https://doi.org/10.1002/ddr.21611

10. Discovery of novel phosphatidylcholine-specific phospholipase C drug-like inhibitors as potential anticancer agents

By: Eurtivong, C., Pilkington, L. I., van Rensburg, M., White, R. M., Brar, H. K., Rees, S., Paulin, E. K., Xu, C. S., Sharma, N., Leung, I. K. H., Leung, E., Barker, D., and Reynisson, J.
European Journal of Medicinal Chemistry
Vol.: 187
No.:
Page:
Published: 2020
doi: https://doi.org/10.1016/j.ejmech.2019.111919

11. Draft Genome Sequence of Diaporthe sp. Strain HANT25, an Endophytic Fungus Producing Mycoepoxydiene

By: Tulsook, K., Isarangkul, D., Sriubolmas, N., Kittakoop, P., and Wiyakrutta, S.
Microbiol Resour Announc
Vol.: 9
No.: 36
Page:
Published: 2020
doi: https://doi.org/10.1128/MRA.00805-20

12. First Draft Genome Sequence of Thermophilic Laceyella tengchongensis BKK01, Isolated from Municipal Solid Waste in Thailand

By: Wachiralurpan, S., Ruangsuj, P., Yamprayoonswat, W., Sopha, P., Jumpathong, W., Sittihan, S., Kanjanavas, P., Areekit, S., Chansiri, K., Chauyrod, K., and Yasawong, M.
Microbiology resource announcements
Vol.: 9
No.: 37
Page: 2
Published: 2020
doi: https://doi.org/10.1128/mra.00798-20

13. Functionalization at C2, C3, and C4 of quinolines: Discovery of water-soluble betaine dyes of C3 quinolinium derivatives with solvatochromic and pH-sensitive properties

By: Sangher, S., Kesornpun, C., Aree, T., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Dyes and Pigments
Vol.: 178
No.:
Page:
Published: 2020
doi: https://doi.org/10.1016/j.dyepig.2020.108341

14. Metal-Free, One-Pot Cascade Annulation of 2-Pyrones in Water for the Synthesis of Peptidomimetics

By: Disadee, W., Lekky, A., and Ruchirawat, S.
Journal of Organic Chemistry
Vol.: 85
No.: 4
Page: 1802-1822
Published: 2020
doi: https://doi.org/10.1021/acs.joc.9b01856

15. Molecular dynamics, MM/PBSA and in vitro validation of a novel quinazoline-based EGFR tyrosine kinase inhibitor identified using structure-based in silico screening

By: Ornnork, N., Kiriwan, D., Lirdprapamongkol, K., Choowongkomon, K., Svasti, J., and Eurtivong, C.
Journal of Molecular Graphics and Modelling
Vol.: 99
No.:
Page:
Published: 2020
doi: https://doi.org/10.1016/j.jmgm.2020.107639

16. Nickel Nanoparticle Catalyzed Mono- and Di-Reductions of gem-Dibromocyclopropanes Under Mild, Aqueous Micellar Conditions

By: Wood, A. B., Cortes-Clerget, M., Kincaid, J. R. A., Akkachairin, B., Singhania, V., Gallou, F., and Lipshutz, B. H.
Angew Chem Int Ed Engl
Vol.:
No.:
Page:
Published: 2020
doi: https://doi.org/10.1002/anie.202006162

17. Rapid synthesis of mycobacterial mannan polysaccharide with alkyne terminated linker

By: Bunthitsakda, W., Ruchirawat, S., and Boonyarattanakalin, S.
Suranaree Journal of Science and Technology
Vol.: 27
No.: 1
Page: 9
Published: 2020
doi:

18. Synthesis and antitumor activity of bis(arylsulfonyl)dihydroimidazolinone derivatives

By: Sittihan, S., Jumpathong, W., Sopha, P., and Ruchirawat, S.
Bioorganic and Medicinal Chemistry Letters
Vol.: 30
No.: 1
Page:
Published: 2020
doi: https://doi.org/10.1016/j.bmcl.2019.126776

19. Synthesis and neuroprotective effects of novel chalcone-triazole hybrids

By: Sooknual, P., Pingaew, R., Phopin, K., Ruankham, W., Prachayasittikul, S., Ruchirawat, S., and Prachayasittikul, V.
Bioorganic Chemistry
Vol.: 105
No.:
Page:
Published: 2020
doi: https://doi.org/10.1016/j.bioorg.2020.104384

20. Synthesis of 4-Acylchromene via Highly Chemoselective Iodine-Catalyzed Cyclization of Alkynylarylether Dimethylacetals

By: Rodphon, W., Thongsornkleeb, C., Tummatorn, J., and Ruchirawat, S.
Chemistry-an Asian Journal
Vol.: 15
No.: 21
Page: 3475-3486
Published: 2020
doi: https://doi.org/10.1002/asia.202000994

21. Synthesis of neocryptolepines and carbocycle-fused quinolines and evaluation of their anticancer and antiplasmodial activities

By: Akkachairin, B., Rodphon, W., Reamtong, O., Mungthin, M., Tummatorn, J., Thongsornkleeb, C., and Ruchirawat, S.
Bioorganic Chemistry
Vol.: 98
No.:
Page:
Published: 2020
doi: https://doi.org/10.1016/j.bioorg.2020.103732

22. Synthesis, cytotoxicity evaluation, and molecular modeling studies of 2,N10-substituted acridones as DNA-intercalating agents

By: Khunnawutmanotham, N., Jumpathong, W., Eurtivong, C., Chimnoi, N., and Techasakul, S.
Journal of Chemical Research
Vol.: 44
No.: 7-8
Page: 410-425
Published: 2020
doi: https://doi.org/10.1177/1747519820902674

23. Transition-Metal-Catalyzed Suzuki-Miyaura-Type Cross-Coupling Reactions of pi-Activated Alcohols

By: Akkarasamiyo, S., Ruchirawat, S., Ploypradith, P., and Samec, J. S. M.
Synthesis-Stuttgart
Vol.: 52
No.: 5
Page: 645-659
Published: 2020
doi: https://doi.org/10.1055/s-0039-1690740

24. UHPLC-ESI-QTOF-MS/MS-Based Molecular Networking Guided Isolation and Dereplication of Antibacterial and Antifungal Constituents of Ventilago denticulata

By: Azizah, M., Pripdeevech, P., Thongkongkaew, T., Mahidol, C., Ruchirawat, S., and Kittakoop, P.
Antibiotics (Basel)
Vol.: 9
No.: 9
Page:
Published: 2020
doi: https://doi.org/10.3390/antibiotics9090606